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Fibrinolytic once daily

University of North Carolina, Chapel Hill · FDA-approved active Small molecule

Fibrinolytic agents dissolve blood clots by activating plasminogen to plasmin, which breaks down fibrin in thrombi.

Fibrinolytic agents dissolve blood clots by activating plasminogen to plasmin, which breaks down fibrin in thrombi. Used for Acute myocardial infarction, Acute ischemic stroke, Pulmonary embolism.

At a glance

Generic nameFibrinolytic once daily
Also known asonce daily lytics, tPA once daily
SponsorUniversity of North Carolina, Chapel Hill
Drug classFibrinolytic agent / Thrombolytic
TargetPlasminogen / Fibrin
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Fibrinolytic drugs work by converting the inactive zymogen plasminogen into its active form, plasmin, a serine protease that degrades fibrin—the structural protein that stabilizes blood clots. This mechanism enables dissolution of existing thrombi in conditions such as acute myocardial infarction, acute ischemic stroke, and pulmonary embolism. Once-daily formulation suggests a modified-release or long-acting variant designed to improve dosing convenience.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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