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Fenoldopam mesilate

IRCCS Policlinico S. Donato · FDA-approved active Small molecule

Fenoldopam mesilate is a selective dopamine-1 (DA1) receptor agonist that causes vasodilation and increases renal blood flow.

Fenoldopam mesilate is a selective dopamine-1 (DA1) receptor agonist that causes vasodilation and increases renal blood flow. Used for Acute hypertension in hospitalized patients, Hypertensive crisis.

At a glance

Generic nameFenoldopam mesilate
Also known asCorlopam
SponsorIRCCS Policlinico S. Donato
Drug classDopamine-1 receptor agonist
TargetDopamine-1 (DA1) receptor
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Fenoldopam selectively binds to dopamine-1 receptors on vascular smooth muscle and renal vasculature, leading to peripheral and renal vasodilation. This results in decreased systemic vascular resistance, lowered blood pressure, and improved renal perfusion. It is used primarily for acute hypertension management in hospital settings.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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