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Fatty Acids, Unsaturated

Wroclaw Medical University · Phase 3 active Small molecule

Unsaturated fatty acids modulate inflammatory pathways and cellular membrane composition to reduce cardiovascular and metabolic dysfunction.

Unsaturated fatty acids modulate inflammatory pathways and cellular membrane composition to reduce cardiovascular and metabolic dysfunction. Used for Hypertriglyceridemia, Cardiovascular disease prevention, Metabolic syndrome.

At a glance

Generic nameFatty Acids, Unsaturated
Also known asOmegaRegen, Esters of Unsaturated Fatty Acids, EFA
SponsorWroclaw Medical University
Drug classLipid therapeutic / Nutraceutical
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

Unsaturated fatty acids, particularly omega-3 and omega-6 polyunsaturated fatty acids, integrate into cell membranes and serve as precursors for bioactive lipid mediators (e.g., prostaglandins, resolvins) that regulate inflammation and immune responses. They also improve lipid profiles, reduce triglycerides, and enhance endothelial function through multiple signaling pathways including GPR120 and PPAR activation.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results