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Eylea® (Aflibercept)
Aflibercept is a soluble decoy receptor that binds and neutralizes vascular endothelial growth factor (VEGF) and placental growth factor (PlGF) to inhibit abnormal blood vessel growth in the eye.
Aflibercept is a soluble decoy receptor that binds and neutralizes vascular endothelial growth factor (VEGF) and placental growth factor (PlGF) to inhibit abnormal blood vessel growth in the eye. Used for Wet age-related macular degeneration (wAMD), Diabetic macular edema (DME), Macular edema following retinal vein occlusion (RVO).
At a glance
| Generic name | Eylea® (Aflibercept) |
|---|---|
| Sponsor | Alvotech Swiss AG |
| Drug class | VEGF inhibitor / Soluble decoy receptor |
| Target | VEGF-A, VEGF-B, PlGF (Placental Growth Factor) |
| Modality | Small molecule |
| Therapeutic area | Ophthalmology |
| Phase | Phase 3 |
Mechanism of action
Aflibercept functions as a fusion protein combining VEGF-binding domains from VEGF receptors 1 and 2 with the Fc portion of human IgG1. By sequestering circulating VEGF and PlGF, it prevents these growth factors from activating their endogenous receptors on endothelial cells, thereby reducing pathological neovascularization and vascular permeability in retinal diseases. This mechanism is particularly effective in wet age-related macular degeneration, diabetic macular edema, and retinal vein occlusion.
Approved indications
- Wet age-related macular degeneration (wAMD)
- Diabetic macular edema (DME)
- Macular edema following retinal vein occlusion (RVO)
- Diabetic retinopathy
Common side effects
- Conjunctival hemorrhage
- Eye pain
- Floaters
- Intraocular pressure elevation
- Endophthalmitis
- Retinal detachment
Key clinical trials
- A Clinical Trial of EYE201/MK-8748 in People With Macular Degeneration (MK-8748-003) (PHASE2, PHASE3)
- 4D-150 in Patients With Macular Neovascularization Secondary to Age-Related Macular Degeneration (PHASE3)
- A Clinical Study of QL1207H Injection Versus Aflibercept for Neovascular Age-related Macular Degeneration (PHASE3)
- A Clinical Trial of EYE201/MK-8748 in People With Macular Degeneration (MK-8748-002) (PHASE2, PHASE3)
- Single Intravitreal (IVT) Injection of 4D-150 in Patients With Macular Neovascularization Secondary to Age-Related Macular Degeneration (PHASE3)
- A Study to Test Whether BI 764524 Helps People With an Eye Condition Called Diabetic Retinopathy (PHASE2)
- Real-Life Clinical Outcomes of Aflibercept Biosimilar MY-1701P in the Treatment of Exudative Age-Related Macular Degeneration
- Comparison of Rapid Aflibercept and Brolucizumab T&E in wAMD (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |