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Estrace® Vaginal Cream USP, 0.01%

Actavis Inc. · Phase 3 active Small molecule

Estrace® Vaginal Cream USP, 0.01% is a Estrogen replacement therapy (local/vaginal) Small molecule drug developed by Actavis Inc.. It is currently in Phase 3 development for Vaginal atrophy and urogenital symptoms associated with menopause, Atrophic vaginitis.

Estrace vaginal cream delivers estradiol directly to vaginal tissue to restore estrogen levels and relieve symptoms of vaginal atrophy and urogenital aging.

Estrace vaginal cream delivers estradiol directly to vaginal tissue to restore estrogen levels and relieve symptoms of vaginal atrophy and urogenital aging. Used for Vaginal atrophy and urogenital symptoms associated with menopause, Atrophic vaginitis.

At a glance

Generic nameEstrace® Vaginal Cream USP, 0.01%
SponsorActavis Inc.
Drug classEstrogen replacement therapy (local/vaginal)
TargetEstrogen receptor alpha (ERα) and estrogen receptor beta (ERβ)
ModalitySmall molecule
Therapeutic areaGynecology / Menopause
PhasePhase 3

Mechanism of action

Estradiol is a bioidentical estrogen that binds to estrogen receptors in the vaginal epithelium, promoting cellular proliferation, increasing vaginal blood flow, and restoring vaginal moisture and elasticity. This local hormone replacement therapy alleviates symptoms such as vaginal dryness, dyspareunia, and urinary discomfort associated with menopause or estrogen deficiency.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Estrace® Vaginal Cream USP, 0.01%

What is Estrace® Vaginal Cream USP, 0.01%?

Estrace® Vaginal Cream USP, 0.01% is a Estrogen replacement therapy (local/vaginal) drug developed by Actavis Inc., indicated for Vaginal atrophy and urogenital symptoms associated with menopause, Atrophic vaginitis.

How does Estrace® Vaginal Cream USP, 0.01% work?

Estrace vaginal cream delivers estradiol directly to vaginal tissue to restore estrogen levels and relieve symptoms of vaginal atrophy and urogenital aging.

What is Estrace® Vaginal Cream USP, 0.01% used for?

Estrace® Vaginal Cream USP, 0.01% is indicated for Vaginal atrophy and urogenital symptoms associated with menopause, Atrophic vaginitis.

Who makes Estrace® Vaginal Cream USP, 0.01%?

Estrace® Vaginal Cream USP, 0.01% is developed by Actavis Inc. (see full Actavis Inc. pipeline at /company/actavis-inc).

What drug class is Estrace® Vaginal Cream USP, 0.01% in?

Estrace® Vaginal Cream USP, 0.01% belongs to the Estrogen replacement therapy (local/vaginal) class. See all Estrogen replacement therapy (local/vaginal) drugs at /class/estrogen-replacement-therapy-local-vaginal.

What development phase is Estrace® Vaginal Cream USP, 0.01% in?

Estrace® Vaginal Cream USP, 0.01% is in Phase 3.

What are the side effects of Estrace® Vaginal Cream USP, 0.01%?

Common side effects of Estrace® Vaginal Cream USP, 0.01% include Vaginal irritation or burning, Headache, Breast tenderness, Vaginal discharge.

What does Estrace® Vaginal Cream USP, 0.01% target?

Estrace® Vaginal Cream USP, 0.01% targets Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) and is a Estrogen replacement therapy (local/vaginal).

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