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ergocalciferol (vitamin D2)

Atlanta VA Medical Center · FDA-approved active Small molecule

Ergocalciferol (vitamin D2) is converted in the body to its active form, which binds to the vitamin D receptor to regulate calcium and phosphate homeostasis and support bone health and immune function.

Ergocalciferol (vitamin D2) is converted in the body to its active form, which binds to the vitamin D receptor to regulate calcium and phosphate homeostasis and support bone health and immune function. Used for Vitamin D deficiency, Hypoparathyroidism, Rickets.

At a glance

Generic nameergocalciferol (vitamin D2)
Also known asD2
SponsorAtlanta VA Medical Center
Drug classVitamin D supplement
TargetVitamin D receptor (VDR)
ModalitySmall molecule
Therapeutic areaEndocrinology / Bone Health
PhaseFDA-approved

Mechanism of action

Ergocalciferol is a plant-derived form of vitamin D that undergoes hydroxylation in the liver and kidneys to form the active metabolite calcitriol. This active form binds to the vitamin D receptor (VDR), a nuclear receptor that modulates gene expression to increase intestinal calcium absorption, regulate serum calcium and phosphate levels, and support bone mineralization. Additionally, vitamin D receptor signaling plays important roles in immune cell differentiation and function.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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