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elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil

Fundacion Clinic per a la Recerca Biomédica · FDA-approved active Small molecule

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is a Antiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors) Small molecule drug developed by Fundacion Clinic per a la Recerca Biomédica. It is currently FDA-approved for HIV-1 infection in treatment-naïve and treatment-experienced adults. Also known as: (Stribild).

This fixed-dose combination inhibits HIV integrase, protease, and reverse transcriptase while blocking viral entry, suppressing HIV replication through multiple mechanisms.

This fixed-dose combination inhibits HIV integrase, protease, and reverse transcriptase while blocking viral entry, suppressing HIV replication through multiple mechanisms. Used for HIV-1 infection in treatment-naïve and treatment-experienced adults.

At a glance

Generic nameelvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil
Also known as(Stribild)
SponsorFundacion Clinic per a la Recerca Biomédica
Drug classAntiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors)
TargetHIV integrase, CYP3A4, HIV reverse transcriptase
ModalitySmall molecule
Therapeutic areaInfectious Disease / Virology
PhaseFDA-approved

Mechanism of action

Elvitegravir is an integrase strand transfer inhibitor that prevents HIV DNA from integrating into the host genome. Cobicistat is a pharmacokinetic booster that inhibits CYP3A4, enhancing elvitegravir levels. Emtricitabine and tenofovir disoproxil are nucleoside/nucleotide reverse transcriptase inhibitors that block viral RNA-dependent DNA polymerase, together providing potent antiretroviral activity against HIV-1.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

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Frequently asked questions about elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil

What is elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is a Antiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors) drug developed by Fundacion Clinic per a la Recerca Biomédica, indicated for HIV-1 infection in treatment-naïve and treatment-experienced adults.

How does elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil work?

This fixed-dose combination inhibits HIV integrase, protease, and reverse transcriptase while blocking viral entry, suppressing HIV replication through multiple mechanisms.

What is elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil used for?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is indicated for HIV-1 infection in treatment-naïve and treatment-experienced adults.

Who makes elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is developed and marketed by Fundacion Clinic per a la Recerca Biomédica (see full Fundacion Clinic per a la Recerca Biomédica pipeline at /company/fundacion-clinic-per-a-la-recerca-biom-dica).

Is elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil also known as anything else?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is also known as (Stribild).

What drug class is elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil in?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil belongs to the Antiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors) class. See all Antiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors) drugs at /class/antiretroviral-combination-integrase-inhibitor-pharmacokinetic-booster-nucleoside-nucleotide-reverse-transcriptase-inhibitors.

What development phase is elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil in?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil is FDA-approved (marketed).

What are the side effects of elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil?

Common side effects of elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil include Nausea, Diarrhea, Headache, Elevated creatinine, Rash.

What does elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil target?

elvitegravir/cobicistat/emtricitabine/Tenofovir-Disoproxil targets HIV integrase, CYP3A4, HIV reverse transcriptase and is a Antiretroviral combination (integrase inhibitor + pharmacokinetic booster + nucleoside/nucleotide reverse transcriptase inhibitors).

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