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Jemperli (DOSTARLIMAB)
Dostarlimab-gxly binds to PD-1 and blocks its interaction with PD-L1 and PD-L2, enhancing the immune response against tumors.
Jemperli (Dostarlimab) is a programmed death receptor-1 (PD-1) blocking antibody developed by GlaxoSmithKline. It works by blocking the PD-1 receptor on immune cells, allowing them to recognize and attack cancer cells. Jemperli is approved for the treatment of recurrent or advanced endometrial cancer. It is a patented product, and its commercial status is owned by GlaxoSmithKline. Key safety considerations include immune-mediated adverse reactions and gastrointestinal toxicity.
At a glance
| Generic name | DOSTARLIMAB |
|---|---|
| Sponsor | GSK |
| Drug class | Programmed Death Receptor-1 Blocking Antibody [EPC] |
| Target | PD-1 |
| Modality | Monoclonal antibody |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
| First approval | 2021 |
| Annual revenue | 800 |
Mechanism of action
Dostarlimab-gxly works by binding to the PD-1 receptor on T cells, preventing it from interacting with its ligands PD-L1 and PD-L2. This blockage releases the inhibition of T-cell activity, allowing the immune system to better recognize and attack tumor cells.
Approved indications
- Recurrent or advanced endometrial cancer
Common side effects
- Fatigue
- Nausea
- Diarrhea
- Anemia
- Constipation
- Decreased lymphocytes
- Decreased sodium
- Increased alkaline phosphatase
- Decreased albumin
- Sepsis
- Acute kidney injury
- Urinary tract infection
Key clinical trials
- Combination Niraparib and Dostarlimab Therapy for Recurrent or Persistent Uterine Serous Carcinoma (PHASE2)
- A Study of Neoadjuvant Dostarlimab Plus Capecitabine Plus Oxaliplatin (CAPEOX) Vs CAPEOX With Previously Untreated T4N0 or Stage III Mismatch Repair Proficient (MMRp)/Microsatellite Stable (MSS) Colon Cancer (PHASE2)
- First-Time-in-Human Study of GSK4381562 in Participants With Advanced Solid Tumors (PHASE1)
- Short-term Fasting Prior to PD-1/PD-L1 Inhibitor Therapy for of Advanced or Metastatic Skin Malignancy (PHASE1)
- I-SPY TRIAL: Neoadjuvant and Personalized Adaptive Novel Agents to Treat Breast Cancer (PHASE2)
- Phase I Trial Testing the Safety and Tolerability of Chemoradiation Followed by Chemotherapy + Dostarlimab for Stage IIIC, Node Positive, Endometrial Cancer (PHASE1)
- A Comprehensive Multiomic Biomarker Evaluation Across Two Single-arm Cohorts to Elucidate Mechanisms of Response and Resistance in Recurrent/Metastatic (R/M) Head and Neck Squamous Cell Carcinoma (HNSCC) (PHASE2)
- Phase II Study of Neoadjuvant Dostarlimab in Patients With Untreated T3-4N0-2 or Stage III pMMR/MSS Resectable Colon Cancer (PHASE2)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
| SEC EDGAR | Revenue + earnings |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Jemperli CI brief — competitive landscape report
- Jemperli updates RSS · CI watch RSS
- GSK portfolio CI