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Motilium (domperidone)

Johnson & Johnson (Janssen) · FDA-approved approved Small molecule Quality 35/100

Domperidone (Motilium) is a peripheral dopamine antagonist prokinetic developed by Janssen. Widely available globally but NOT approved in the US. Preferred over metoclopramide for avoiding CNS side effects.

At a glance

Generic namedomperidone
Also known asMotilium
SponsorJohnson & Johnson (Janssen)
Drug classProkinetic agent / Antiemetic
TargetAldehyde oxidase, Multidrug and toxin extrusion protein 1, Multidrug and toxin extrusion protein 2
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved
First approval1978-01-01 (Belgium)

Approved indications

Common side effects

No common side effects on file.

Key clinical trials

Primary sources

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SourceUsed for
FDA labelMechanism, indications, dosing, boxed warnings, drug interactions
ClinicalTrials.govTrial enrolment, design, endpoints, results