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Dolutegravir/lamivudine/abacavir

Azienda Ospedaliera Universitaria Senese · Phase 3 active Small molecule

Dolutegravir/lamivudine/abacavir is a Antiretroviral combination (INSTI + NRTI backbone) Small molecule drug developed by Azienda Ospedaliera Universitaria Senese. It is currently in Phase 3 development for HIV-1 infection in treatment-naïve and treatment-experienced adults, HIV-1 infection in adolescents and children (age-appropriate formulations). Also known as: Triumeq.

This combination of three antiretroviral drugs inhibits HIV replication by blocking integrase and reverse transcriptase enzymes while providing nucleoside backbone coverage.

This combination of three antiretroviral drugs inhibits HIV replication by blocking integrase and reverse transcriptase enzymes while providing nucleoside backbone coverage. Used for HIV-1 infection in treatment-naïve and treatment-experienced adults, HIV-1 infection in adolescents and children (age-appropriate formulations).

At a glance

Generic nameDolutegravir/lamivudine/abacavir
Also known asTriumeq
SponsorAzienda Ospedaliera Universitaria Senese
Drug classAntiretroviral combination (INSTI + NRTI backbone)
TargetHIV integrase, HIV reverse transcriptase
ModalitySmall molecule
Therapeutic areaInfectious Disease / Virology
PhasePhase 3

Mechanism of action

Dolutegravir is an integrase strand transfer inhibitor (INSTI) that prevents HIV DNA from integrating into the host genome. Lamivudine and abacavir are nucleoside reverse transcriptase inhibitors (NRTIs) that block reverse transcriptase, preventing conversion of viral RNA to DNA. Together, they provide complementary mechanisms to suppress HIV replication at multiple steps.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Dolutegravir/lamivudine/abacavir

What is Dolutegravir/lamivudine/abacavir?

Dolutegravir/lamivudine/abacavir is a Antiretroviral combination (INSTI + NRTI backbone) drug developed by Azienda Ospedaliera Universitaria Senese, indicated for HIV-1 infection in treatment-naïve and treatment-experienced adults, HIV-1 infection in adolescents and children (age-appropriate formulations).

How does Dolutegravir/lamivudine/abacavir work?

This combination of three antiretroviral drugs inhibits HIV replication by blocking integrase and reverse transcriptase enzymes while providing nucleoside backbone coverage.

What is Dolutegravir/lamivudine/abacavir used for?

Dolutegravir/lamivudine/abacavir is indicated for HIV-1 infection in treatment-naïve and treatment-experienced adults, HIV-1 infection in adolescents and children (age-appropriate formulations).

Who makes Dolutegravir/lamivudine/abacavir?

Dolutegravir/lamivudine/abacavir is developed by Azienda Ospedaliera Universitaria Senese (see full Azienda Ospedaliera Universitaria Senese pipeline at /company/azienda-ospedaliera-universitaria-senese).

Is Dolutegravir/lamivudine/abacavir also known as anything else?

Dolutegravir/lamivudine/abacavir is also known as Triumeq.

What drug class is Dolutegravir/lamivudine/abacavir in?

Dolutegravir/lamivudine/abacavir belongs to the Antiretroviral combination (INSTI + NRTI backbone) class. See all Antiretroviral combination (INSTI + NRTI backbone) drugs at /class/antiretroviral-combination-insti-nrti-backbone.

What development phase is Dolutegravir/lamivudine/abacavir in?

Dolutegravir/lamivudine/abacavir is in Phase 3.

What are the side effects of Dolutegravir/lamivudine/abacavir?

Common side effects of Dolutegravir/lamivudine/abacavir include Diarrhea, Nausea, Headache, Insomnia, Hypersensitivity reaction (abacavir), Hepatotoxicity.

What does Dolutegravir/lamivudine/abacavir target?

Dolutegravir/lamivudine/abacavir targets HIV integrase, HIV reverse transcriptase and is a Antiretroviral combination (INSTI + NRTI backbone).

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