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Dexlansoprazole MR QD
Dexlansoprazole MR QD is a Proton pump inhibitor (PPI) Small molecule drug developed by Takeda. It is currently in Phase 3 development for Gastroesophageal reflux disease (GERD), Healing of erosive esophagitis, Maintenance of healed erosive esophagitis. Also known as: TAK-390, T-168390, TAK-390MR, Kapidex.
Dexlansoprazole is a proton pump inhibitor that suppresses gastric acid secretion by irreversibly blocking the H+/K+-ATPase enzyme in parietal cells.
Dexlansoprazole is a proton pump inhibitor that suppresses gastric acid secretion by irreversibly blocking the H+/K+-ATPase enzyme in parietal cells. Used for Gastroesophageal reflux disease (GERD), Healing of erosive esophagitis, Maintenance of healed erosive esophagitis.
At a glance
| Generic name | Dexlansoprazole MR QD |
|---|---|
| Also known as | TAK-390, T-168390, TAK-390MR, Kapidex, Dexilant |
| Sponsor | Takeda |
| Drug class | Proton pump inhibitor (PPI) |
| Target | H+/K+-ATPase |
| Modality | Small molecule |
| Therapeutic area | Gastroenterology |
| Phase | Phase 3 |
Mechanism of action
Dexlansoprazole is the active R-enantiomer of lansoprazole, a proton pump inhibitor (PPI). It binds to and inactivates the hydrogen-potassium adenosine triphosphatase (H+/K+-ATPase) pump on the secretory surface of gastric parietal cells, preventing the final step of gastric acid production. The modified-release (MR) formulation provides dual-peak plasma concentrations to maintain acid suppression throughout the day with once-daily dosing.
Approved indications
- Gastroesophageal reflux disease (GERD)
- Healing of erosive esophagitis
- Maintenance of healed erosive esophagitis
Common side effects
- Headache
- Diarrhea
- Abdominal pain
- Nausea
- Upper respiratory tract infection
Key clinical trials
- Dexlansoprazole MR-Based Concomitant Quadruple Therapy (NA)
- Safety and Quality of Life Study of Dexlansoprazole Modified Release Formulation to Treat Heartburn (PHASE3)
- Efficacy and Safety of Dexlansoprazole MR Compared to Placebo on Maintaining Healing in Subjects With Healed Erosive Esophagitis (PHASE3)
- Efficacy and Safety of Dexlansoprazole MR and Lansoprazole on Healing of Erosive Esophagitis (PHASE3)
- Comparison of Dexlansoprazole MR to Placebo on the Ability to Maintain Healing in Subjects With Healed Erosive Esophagitis (PHASE3)
- Efficacy of Dexlansoprazole MR on Heartburn Control in Participants Previously Receiving Twice Daily Proton Pump Inhibitor Therapy (PHASE3)
- Efficacy and Safety of Dexlansoprazole MR and Lansoprazole on Healing of Erosive Esophagitis (PHASE3)
- Efficacy and Safety of Dexlansoprazole MR on Maintaining Healing in Subjects With Healed Erosive Esophagitis (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Dexlansoprazole MR QD CI brief — competitive landscape report
- Dexlansoprazole MR QD updates RSS · CI watch RSS
- Takeda portfolio CI
Frequently asked questions about Dexlansoprazole MR QD
What is Dexlansoprazole MR QD?
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What is Dexlansoprazole MR QD used for?
Who makes Dexlansoprazole MR QD?
Is Dexlansoprazole MR QD also known as anything else?
What drug class is Dexlansoprazole MR QD in?
What development phase is Dexlansoprazole MR QD in?
What are the side effects of Dexlansoprazole MR QD?
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Related
- Drug class: All Proton pump inhibitor (PPI) drugs
- Target: All drugs targeting H+/K+-ATPase
- Manufacturer: Takeda — full pipeline
- Therapeutic area: All drugs in Gastroenterology
- Indication: Drugs for Gastroesophageal reflux disease (GERD)
- Indication: Drugs for Healing of erosive esophagitis
- Indication: Drugs for Maintenance of healed erosive esophagitis
- Also known as: TAK-390, T-168390, TAK-390MR, Kapidex, Dexilant
- Compare: Dexlansoprazole MR QD vs similar drugs
- Pricing: Dexlansoprazole MR QD cost, discount & access