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Desflurane with remifentanil

Chung-Ang University Hosptial, Chung-Ang University College of Medicine · FDA-approved active Small molecule

Desflurane is a volatile anesthetic that depresses the central nervous system, while remifentanil is an opioid agonist that provides analgesia and enhances anesthesia.

Desflurane is a volatile anesthetic that depresses the central nervous system, while remifentanil is an opioid agonist that provides analgesia and enhances anesthesia. Used for General anesthesia for surgical procedures.

At a glance

Generic nameDesflurane with remifentanil
Also known asdesflurane with remifetanil group
SponsorChung-Ang University Hosptial, Chung-Ang University College of Medicine
Drug classVolatile anesthetic with opioid analgesic
TargetGABA receptors (desflurane); mu-opioid receptors (remifentanil)
ModalitySmall molecule
Therapeutic areaAnesthesiology
PhaseFDA-approved

Mechanism of action

Desflurane works by enhancing inhibitory GABAergic neurotransmission and inhibiting excitatory glutamatergic signaling in the brain, producing unconsciousness and amnesia. Remifentanil binds to mu-opioid receptors in the central nervous system to provide rapid-onset analgesia and potentiate the anesthetic effect. Together, this combination provides balanced general anesthesia with rapid emergence due to remifentanil's ultra-short half-life.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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