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Demethylchlortetracycline (DEMECLOCYCLINE)
Demethylchlortetracycline (generic name: DEMECLOCYCLINE) is a Tetracycline-class Antimicrobial Small molecule drug developed by Pfizer. It is currently FDA-approved (first approved 1960) for Actinomycotic infection, Acute bacterial sinusitis, Acute gonococcal cervicitis.
Demethylchlortetracycline (DEMECLOCYCLINE) is a tetracycline-class antimicrobial drug originally developed by Lederle and currently owned by the same company. It targets the estrogen receptor beta and has been FDA-approved since 1960 for various bacterial infections, including actinomycotic infections, acute bacterial sinusitis, and anthrax. The drug is a small molecule with a half-life of 12 hours and bioavailability of 66%. It is off-patent and has multiple generic manufacturers. Key safety considerations include its potential to interact with other medications and affect liver function.
At a glance
| Generic name | DEMECLOCYCLINE |
|---|---|
| Sponsor | Pfizer |
| Drug class | Tetracycline-class Antimicrobial |
| Target | Estrogen receptor beta |
| Modality | Small molecule |
| Therapeutic area | Immunology |
| Phase | FDA-approved |
| First approval | 1960 |
Approved indications
- Actinomycotic infection
- Acute bacterial sinusitis
- Acute gonococcal cervicitis
- Acute gonococcal endometritis
- Acute gonococcal urethritis
- Anthrax
- Bronchitis
- Brucellosis
- Chancroid
- Gingivostomatitis
- Gonorrhea
- Gonorrhea of pharynx
- Gonorrhea of rectum
- Granuloma inguinale
- Haemophilus Influenzae Acute Otitis Media
- Haemophilus Influenzae Pharyngitis
- Inclusion conjunctivitis
- Infection due to Staphylococcus aureus
- Infection of skin AND/OR subcutaneous tissue
- Infective otitis media
Common side effects
- Hepatitis
- Liver failure
- Pancreatitis
- Hepatic toxicity
- Acute renal failure
- Rise in BUN
- Nephrogenic diabetes insipidus
- Pseudotumor cerebri (benign intracranial hypertension)
- Bulging fontanels
- Anaphylaxis
- Anaphylactoid purpura
- Pericarditis
Key clinical trials
- Patients Response to Early Switch To Oral:Osteomyelitis Study (EARLY_PHASE1)
- Bone Histomorphometry in Postmenopausal Men and Women With Osteoarthritis Undergoing Total Hip Replacement (PHASE4)
- The Impact of Parathyroid Hormone (PTH) on Craniofacial Osseous Regeneration in Bone (PHASE2)
- Demeclocycline Fluorescence for Intraoperative Delineation Brain Tumors (PHASE1)
- Effects of Teriparatide or Denosumab on Bone in Postmenopausal Women With Osteoporosis (PHASE4)
- S0307A, Long-Term Bone Quality in Women With Breast Cancer Enrolled on Clinical Trial SWOG-S0307
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Demethylchlortetracycline CI brief — competitive landscape report
- Demethylchlortetracycline updates RSS · CI watch RSS
- Pfizer portfolio CI
Frequently asked questions about Demethylchlortetracycline
What is Demethylchlortetracycline?
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What is the generic name of Demethylchlortetracycline?
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When was Demethylchlortetracycline approved?
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Related
- Drug class: All Tetracycline-class Antimicrobial drugs
- Target: All drugs targeting Estrogen receptor beta
- Manufacturer: Pfizer — full pipeline
- Therapeutic area: All drugs in Immunology
- Indication: Drugs for Actinomycotic infection
- Indication: Drugs for Acute bacterial sinusitis
- Indication: Drugs for Acute gonococcal cervicitis
Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing