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Delamanid in Oral Dosage Form
Delamanid in Oral Dosage Form is a Mycobacterial cell wall synthesis inhibitor Small molecule drug developed by Wits Health Consortium (Pty) Ltd. It is currently in Phase 3 development for Drug-resistant tuberculosis (MDR-TB and XDR-TB), Pulmonary tuberculosis in combination with other anti-tuberculous agents. Also known as: Deltyba.
Delamanid inhibits mycobacterial cell wall synthesis by targeting mycolic acid production, thereby killing Mycobacterium tuberculosis.
Delamanid inhibits mycobacterial cell wall synthesis by targeting mycolic acid production, thereby killing Mycobacterium tuberculosis. Used for Drug-resistant tuberculosis (MDR-TB and XDR-TB), Pulmonary tuberculosis in combination with other anti-tuberculous agents.
At a glance
| Generic name | Delamanid in Oral Dosage Form |
|---|---|
| Also known as | Deltyba |
| Sponsor | Wits Health Consortium (Pty) Ltd |
| Drug class | Mycobacterial cell wall synthesis inhibitor |
| Target | DprE1 (decaprenylphosphoryl-arabinose-1-phosphatase) |
| Modality | Small molecule |
| Therapeutic area | Infectious Disease |
| Phase | Phase 3 |
Mechanism of action
Delamanid is a nitro-aromatic prodrug that is activated by mycobacterial enzymes to form reactive intermediates that inhibit the enzyme DprE1, which is essential for the synthesis of decaprenylphosphoryl-arabinose—a critical precursor for mycolic acid biosynthesis in the mycobacterial cell wall. By disrupting cell wall integrity, delamanid leads to mycobacterial cell death and is particularly effective against drug-resistant tuberculosis strains.
Approved indications
- Drug-resistant tuberculosis (MDR-TB and XDR-TB)
- Pulmonary tuberculosis in combination with other anti-tuberculous agents
Common side effects
- Nausea
- Vomiting
- Abdominal pain
- Headache
- Peripheral neuropathy
- QT prolongation
Key clinical trials
- Pharmacokinetic Study of Antiretroviral Drugs and Related Drugs During and After Pregnancy
- Early Bactericidal Activity, Safety & Tolerability of Oral GSK3036656 in a Dual Combination With Novel and Established Antitubercular Agents, or Standard of Care in Adults With Rifampicin Susceptible Pulmonary Tuberculosis (PHASE2)
- Platform Assessing Regimens and Durations In a Global Multisite Consortium for TB (PHASE2)
- 6 Months of Bedaquiline(BDQ), Delamanid(DLM), Linezolid(LZD) and Levofloxacin(LFX) in RR-TB Patients in Hubei Province (NA)
- PanACEA DElpazolid Dose-finding and COmbination DEvelopment (DECODE) (PHASE2)
- Efficacy and Tolerability of Bedaquiline, Delamanid, Levofloxacin, Linezolid, and Clofazimine to Treat MDR-TB (PHASE2)
- Safety and Efficacy Evaluation of 4-month Regimen of OPC-167832, Delamanid and Bedaquiline in Participants With Drug-Susceptible Pulmonary TB (PHASE2)
- Evaluating Newly Approved Drugs in Combination Regimens for Multidrug-Resistant TB With Fluoroquinolone Resistance (endTB-Q) (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Delamanid in Oral Dosage Form CI brief — competitive landscape report
- Delamanid in Oral Dosage Form updates RSS · CI watch RSS
- Wits Health Consortium (Pty) Ltd portfolio CI
Frequently asked questions about Delamanid in Oral Dosage Form
What is Delamanid in Oral Dosage Form?
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Related
- Drug class: All Mycobacterial cell wall synthesis inhibitor drugs
- Target: All drugs targeting DprE1 (decaprenylphosphoryl-arabinose-1-phosphatase)
- Manufacturer: Wits Health Consortium (Pty) Ltd — full pipeline
- Therapeutic area: All drugs in Infectious Disease
- Indication: Drugs for Drug-resistant tuberculosis (MDR-TB and XDR-TB)
- Indication: Drugs for Pulmonary tuberculosis in combination with other anti-tuberculous agents
- Also known as: Deltyba
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