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Daratumumab/rHuPH20

Masonic Cancer Center, University of Minnesota · Phase 3 active Small molecule

Daratumumab is a monoclonal antibody that targets CD38 on multiple myeloma cells, while rHuPH20 is a recombinant human hyaluronidase that enhances subcutaneous delivery by breaking down hyaluronic acid in the extracellular matrix.

Daratumumab is a monoclonal antibody that targets CD38 on multiple myeloma cells, while rHuPH20 is a recombinant human hyaluronidase that enhances subcutaneous delivery by breaking down hyaluronic acid in the extracellular matrix. Used for Multiple myeloma (subcutaneous formulation in phase 3 development).

At a glance

Generic nameDaratumumab/rHuPH20
Also known asDarzalex
SponsorMasonic Cancer Center, University of Minnesota
Drug classMonoclonal antibody with recombinant human hyaluronidase
TargetCD38
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

Daratumumab binds to CD38, a surface antigen highly expressed on multiple myeloma cells, triggering immune-mediated cell death through antibody-dependent cellular cytotoxicity (ADCC), complement-dependent cytotoxicity (CDC), and antibody-dependent cellular phagocytosis (ADCP). The rHuPH20 enzyme facilitates rapid subcutaneous absorption by temporarily degrading hyaluronic acid in subcutaneous tissue, allowing for faster and more complete drug delivery compared to standard subcutaneous administration.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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