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Daily Vitamin D3

Medical University of South Carolina · FDA-approved active Small molecule

Vitamin D3 (cholecalciferol) is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function.

Vitamin D3 (cholecalciferol) is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function. Used for Vitamin D deficiency prevention and treatment, Support of bone health and calcium homeostasis, Immune function support.

At a glance

Generic nameDaily Vitamin D3
Also known asDaily cholecalciferol
SponsorMedical University of South Carolina
Drug classVitamin/nutritional supplement
TargetVitamin D receptor (VDR)
ModalitySmall molecule
Therapeutic areaNutritional/Metabolic
PhaseFDA-approved

Mechanism of action

Vitamin D3 is a fat-soluble vitamin that undergoes hydroxylation in the liver and kidneys to form the active hormone calcitriol (1,25-dihydroxyvitamin D3). This active metabolite binds to the vitamin D receptor (VDR) in target tissues, promoting intestinal calcium and phosphate absorption, regulating bone mineralization, and modulating immune cell differentiation and function. It plays a critical role in maintaining serum calcium levels and skeletal health.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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