Last reviewed · How we verify

D3 vitamin

Medical University of Lodz · FDA-approved active Small molecule

Vitamin D3 (cholecalciferol) is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function.

Vitamin D3 (cholecalciferol) is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function. Used for Vitamin D deficiency, Hypocalcemia, Osteoporosis prevention and treatment.

At a glance

Generic nameD3 vitamin
Also known asD3 Vitamin ®, supplied by D3 Pharmacy Ltd, D3
SponsorMedical University of Lodz
Drug classVitamin D supplement / Secosteroid
TargetVitamin D receptor (VDR)
ModalitySmall molecule
Therapeutic areaEndocrinology / Bone metabolism / Immunology
PhaseFDA-approved

Mechanism of action

Vitamin D3 is a fat-soluble vitamin that undergoes hydroxylation in the liver and kidneys to form the active hormone calcitriol (1,25-dihydroxyvitamin D3). This active metabolite binds to the vitamin D receptor (VDR) in target tissues, promoting intestinal calcium and phosphate absorption, regulating bone mineralization, and modulating immune cell differentiation and function. It plays a critical role in maintaining serum calcium levels and skeletal health.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape: