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copper histidinate

Sentynl Therapeutics, Inc. · FDA-approved active Small molecule

Copper histidinate provides bioavailable copper to restore deficient copper levels in patients with copper malabsorption or deficiency.

Copper histidinate provides bioavailable copper to restore deficient copper levels in patients with copper malabsorption or deficiency. Used for Copper deficiency due to malabsorption (including Menkes disease and related copper transport disorders).

At a glance

Generic namecopper histidinate
Also known asCUTX-101
SponsorSentynl Therapeutics, Inc.
Drug classTrace element supplement
TargetCopper ion (Cu2+)
ModalitySmall molecule
Therapeutic areaMetabolic/Genetic Disorders
PhaseFDA-approved

Mechanism of action

Copper is an essential trace element required for multiple enzymatic processes including cytochrome c oxidase, lysyl oxidase, and superoxide dismutase. Copper histidinate is a chelate complex that enhances copper absorption in the gastrointestinal tract, allowing systemic copper repletion in patients who cannot adequately absorb dietary copper due to genetic disorders or malabsorption conditions.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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