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Clindamycin + primaquine

McGill University Health Centre/Research Institute of the McGill University Health Centre · FDA-approved active Small molecule

Clindamycin + primaquine is a Antibiotic + antiprotozoal combination Small molecule drug developed by McGill University Health Centre/Research Institute of the McGill University Health Centre. It is currently FDA-approved for Pneumocystis jirovecii pneumonia (PCP) prophylaxis and treatment.

Clindamycin inhibits bacterial protein synthesis while primaquine acts as an antimalarial and antiprotozoal agent, together targeting Pneumocystis jirovecii pneumonia (PCP).

Clindamycin inhibits bacterial protein synthesis while primaquine acts as an antimalarial and antiprotozoal agent, together targeting Pneumocystis jirovecii pneumonia (PCP). Used for Pneumocystis jirovecii pneumonia (PCP) prophylaxis and treatment.

At a glance

Generic nameClindamycin + primaquine
SponsorMcGill University Health Centre/Research Institute of the McGill University Health Centre
Drug classAntibiotic + antiprotozoal combination
TargetBacterial ribosome (clindamycin); protozoal metabolism (primaquine)
ModalitySmall molecule
Therapeutic areaInfectious Disease
PhaseFDA-approved

Mechanism of action

Clindamycin is a lincosamide antibiotic that binds to bacterial ribosomes and inhibits protein synthesis. Primaquine is an 8-aminoquinoline that generates reactive oxygen species within protozoal parasites, disrupting their metabolism. This combination is used to treat PCP, particularly in patients who cannot tolerate trimethoprim-sulfamethoxazole.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Clindamycin + primaquine

What is Clindamycin + primaquine?

Clindamycin + primaquine is a Antibiotic + antiprotozoal combination drug developed by McGill University Health Centre/Research Institute of the McGill University Health Centre, indicated for Pneumocystis jirovecii pneumonia (PCP) prophylaxis and treatment.

How does Clindamycin + primaquine work?

Clindamycin inhibits bacterial protein synthesis while primaquine acts as an antimalarial and antiprotozoal agent, together targeting Pneumocystis jirovecii pneumonia (PCP).

What is Clindamycin + primaquine used for?

Clindamycin + primaquine is indicated for Pneumocystis jirovecii pneumonia (PCP) prophylaxis and treatment.

Who makes Clindamycin + primaquine?

Clindamycin + primaquine is developed and marketed by McGill University Health Centre/Research Institute of the McGill University Health Centre (see full McGill University Health Centre/Research Institute of the McGill University Health Centre pipeline at /company/mcgill-university-health-centre-research-institute-of-the-mcgill-university-heal).

What drug class is Clindamycin + primaquine in?

Clindamycin + primaquine belongs to the Antibiotic + antiprotozoal combination class. See all Antibiotic + antiprotozoal combination drugs at /class/antibiotic-antiprotozoal-combination.

What development phase is Clindamycin + primaquine in?

Clindamycin + primaquine is FDA-approved (marketed).

What are the side effects of Clindamycin + primaquine?

Common side effects of Clindamycin + primaquine include Rash, Nausea, Diarrhea, Hemolytic anemia (in G6PD-deficient patients), Methemoglobinemia.

What does Clindamycin + primaquine target?

Clindamycin + primaquine targets Bacterial ribosome (clindamycin); protozoal metabolism (primaquine) and is a Antibiotic + antiprotozoal combination.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing