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cis-platinum

Peking University Third Hospital · FDA-approved active Small molecule

Cisplatin is a platinum-based chemotherapy agent that forms DNA adducts and cross-links, preventing DNA replication and transcription to induce cancer cell death.

Cisplatin is a platinum-based chemotherapy agent that forms DNA adducts and cross-links, preventing DNA replication and transcription to induce cancer cell death. Used for Metastatic testicular cancer, Metastatic ovarian cancer, Advanced bladder cancer.

At a glance

Generic namecis-platinum
Also known asCisplatin, Cisplantin Injection, cisplatin, Platinol
SponsorPeking University Third Hospital
Drug classPlatinum-based alkylating agent
TargetDNA
ModalitySmall molecule
Therapeutic areaOncology
PhaseFDA-approved

Mechanism of action

Cisplatin enters cancer cells and undergoes aquation to form reactive platinum species that bind to purine bases in DNA, creating intrastrand and interstrand cross-links. These DNA lesions trigger apoptosis and cell cycle arrest, leading to cancer cell death. The drug is non-cell-cycle specific and effective against rapidly dividing cells.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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