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2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine (CHLORPROETHAZINE)

Phase 2 active Small molecule

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine (generic name: CHLORPROETHAZINE) is a chlorproethazine drug. It is currently in Phase 2 development.

Chlorproethazine works by blocking the action of dopamine at the D(3) receptor, which can help regulate various physiological processes.

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine, also known as Chlorproethazine, is a small molecule targeting the D(3) dopamine receptor. It belongs to the chlorproethazine drug class but its commercial status, including patent and generic availability, is unknown. The FDA approval status for Chlorproethazine is also unclear. As a dopamine receptor antagonist, it is likely used to treat conditions related to dopamine dysregulation, but specific approved indications are not available. Further research is needed to understand its pharmacokinetic properties and safety considerations.

Likelihood of approval
15.3% vs 15.3% industry baseline
If approved by FDA: likely 2031–2034
Steps remaining: Phase 3 → NDA/BLA submission
Confidence: Medium
Why this estimate
  • Baseline phase 2 → approval rate +15.3pp
    Industry-wide phase 2 drugs reach approval ~15.3% of the time (BIO/Informa 2023 industry benchmark across all therapeutic areas).
Predicted approval windows by jurisdiction (conditional on FDA approval)
Regulator Country Likely year Lag vs FDA
FDA US 2031–2034
EMA EU 2032–2035 +0.7 yr
MHRA GB 2032–2035 +0.7 yr
Health Canada CA 2032–2036 +0.9 yr
TGA AU 2032–2036 +1.2 yr
PMDA JP 2032–2036 +1.5 yr
NMPA CN 2033–2037 +2.3 yr
MFDS KR 2032–2036 +1.4 yr
CDSCO IN 2032–2037 +1.8 yr
ANVISA BR 2033–2037 +2.3 yr

Hover any row for the lag rationale. Lag estimates are reduced when the drug has FDA Breakthrough or EMA PRIME designation (sponsors file globally in parallel).

Estimate based on the BIO/Informa industry phase transition rates plus per-drug modifiers for therapeutic area, sponsor type, FDA designations, mechanism, and trial design. Per-jurisdiction lags from Tufts CSDD international approval studies. Not investment, clinical or regulatory advice. Methodology: /methodology#likelihood.

At a glance

Generic nameCHLORPROETHAZINE
Drug classchlorproethazine
TargetD(4) dopamine receptor, D(2) dopamine receptor, D(3) dopamine receptor
ModalitySmall molecule
Therapeutic areaOther
PhasePhase 2

Mechanism of action

Imagine dopamine as a key that unlocks a door. The D(3) receptor is like the lock on that door. When dopamine binds to the receptor, it can trigger various effects in the body. Chlorproethazine acts like a lockout device, preventing dopamine from binding to the receptor and thereby reducing its effects.

Approved indications

No approved indications tracked.

Common side effects

No common side effects on file.

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine

What is 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine?

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine (CHLORPROETHAZINE) is a chlorproethazine drug.

How does 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine work?

Chlorproethazine works by blocking the action of dopamine at the D(3) receptor, which can help regulate various physiological processes.

What is the generic name of 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine?

CHLORPROETHAZINE is the generic (nonproprietary) name of 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine.

What drug class is 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine in?

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine belongs to the chlorproethazine class. See all chlorproethazine drugs at /class/chlorproethazine.

What development phase is 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine in?

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine is in Phase 2.

What does 2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine target?

2-Chloro-10-(3-Diethylaminopropyl)Phenothiazine targets D(4) dopamine receptor, D(2) dopamine receptor, D(3) dopamine receptor and is a chlorproethazine.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing