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Chlorhexidine rinse

Universidade Estadual Paulista Júlio de Mesquita Filho · FDA-approved active Small molecule

Chlorhexidine rinse works by disrupting bacterial cell membranes and precipitating bacterial proteins, providing broad-spectrum antimicrobial activity in the oral cavity.

Chlorhexidine rinse works by disrupting bacterial cell membranes and precipitating bacterial proteins, providing broad-spectrum antimicrobial activity in the oral cavity. Used for Gingivitis prevention and treatment, Plaque reduction, Oral antimicrobial rinse.

At a glance

Generic nameChlorhexidine rinse
Also known asDrug prescription, Chlorhexidine, Paroex
SponsorUniversidade Estadual Paulista Júlio de Mesquita Filho
Drug classAntimicrobial oral rinse
TargetBacterial cell membrane and proteins
ModalitySmall molecule
Therapeutic areaOral health / Dentistry
PhaseFDA-approved

Mechanism of action

Chlorhexidine is a cationic biguanide that binds to negatively charged bacterial cell membranes, causing leakage of intracellular contents and cell death. It also denatures bacterial proteins and inhibits bacterial enzymes. The rinse formulation allows direct contact with oral tissues and microorganisms, making it effective for reducing plaque and preventing gingivitis.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results