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Certolizumab Pegol (CZP)

UCB Pharma · FDA-approved active Biologic

Certolizumab pegol is a TNF-alpha inhibitor that binds to and neutralizes tumor necrosis factor-alpha, reducing inflammatory signaling.

Certolizumab pegol is a TNF-alpha inhibitor that binds to and neutralizes tumor necrosis factor-alpha, reducing inflammatory signaling. Used for Rheumatoid arthritis, Crohn's disease, Psoriatic arthritis.

At a glance

Generic nameCertolizumab Pegol (CZP)
Also known asCimzia, CDP870, CZP, Brand Name: Cimzia, UCB product: Certolizumab Pegol (CDP870)
SponsorUCB Pharma
Drug classTNF-alpha inhibitor
TargetTNF-alpha
ModalityBiologic
Therapeutic areaImmunology
PhaseFDA-approved

Mechanism of action

Certolizumab pegol is a pegylated anti-TNF monoclonal antibody fragment that selectively binds to soluble and membrane-bound TNF-alpha, preventing its interaction with TNF receptors. This blocks the inflammatory cascade driven by TNF-alpha, reducing systemic inflammation and immune activation. Unlike full monoclonal antibodies, its smaller size and pegylation provide extended half-life and improved tissue penetration.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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