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Libtayo (CEMIPLIMAB)
Cemiplimab-rwlc binds to PD-1 and blocks its interaction with PD-L1 and PD-L2, enhancing the immune response against tumors.
Libtayo (cemiplimab) is a monoclonal antibody developed by Regeneron Pharmaceuticals, targeting the programmed cell death protein 1 (PD-1). It works by blocking the PD-1 receptor, allowing the immune system to recognize and attack cancer cells. Libtayo is approved to treat various types of cancer, including cervical cancer, basal cell carcinoma, and non-small cell lung cancer. It remains a patented product, and its commercial status is unchanged. Key safety considerations include immune-mediated adverse reactions and potential liver damage.
At a glance
| Generic name | CEMIPLIMAB |
|---|---|
| Sponsor | Regeneron Pharmaceuticals |
| Target | PD-1 |
| Modality | Monoclonal antibody |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
| First approval | 2018 |
| Annual revenue | 1452 |
Mechanism of action
Cemiplimab-rwlc works by binding to the PD-1 receptor on T cells, preventing it from interacting with its ligands PD-L1 and PD-L2. This blockage releases the inhibition of T-cell activity, allowing the immune system to better recognize and attack tumor cells.
Approved indications
- Malignant tumor of cervix
- Metastatic basal cell carcinoma
- Non-small cell lung cancer without mutation in epidermal growth factor receptor
- Nonsmall cell lung cancer without mutation in epidermal growth factor receptor
- Squamous cell carcinoma
Common side effects
- fatigue
- rash
- musculoskeletal pain
- diarrhea
- pruritus
- nausea
Key clinical trials
- PD-1 in Patients With Advanced Basal Cell Carcinoma Who Experienced Progression of Disease on Hedgehog Pathway Inhibitor Therapy, or Were Intolerant of Prior Hedgehog Pathway Inhibitor Therapy (PHASE2)
- Study of REGN2810 in Patients With Advanced Cutaneous Squamous Cell Carcinoma (PHASE2)
- Study of REGN2810 (Anti-PD-1) in Patients With Advanced Malignancies (PHASE1)
- Reduced-dose Carboplatin-doublet-chemotherapy + Cemiplimab vs Cemiplimab Monotherapy in Treatment Naive Older and Frail Patients With Metastatic NSCLC With PD-L1 <50% (PHASE2)
- Testing Whether Cemiplimab (REGN2810) Plus CDX-1140 Given Prior to Surgery Are Better Than Cemiplimab (REGN2810) Alone in Patients With Stage III-IV Head and Neck Cancer (PHASE2)
- Testing the Effectiveness of the Anti-cancer Drug Pidnarulex (CX-5461) in Combination With Another Anti-cancer Drug Cemiplimab (REGN2810), in Treating Refractory Microsatellite Stable Colorectal Cancer (PHASE1,PHASE2)
- A Study of Fianlimab, Cemiplimab, and Ipilimumab in People With Melanoma (PHASE2)
- Study of Adjuvant Cemiplimab Versus Placebo After Surgery and Radiation Therapy in Patients With High Risk Cutaneous Squamous Cell Carcinoma (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
| SEC EDGAR | Revenue + earnings |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Libtayo CI brief — competitive landscape report
- Libtayo updates RSS · CI watch RSS
- Regeneron Pharmaceuticals portfolio CI