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Cefazolin PostOperatively

Aultman Health Foundation · FDA-approved active Small molecule

Cefazolin is a first-generation cephalosporin antibiotic that inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins.

Cefazolin is a first-generation cephalosporin antibiotic that inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins. Used for Surgical site infection prophylaxis (postoperative use), Bacterial infections caused by susceptible organisms.

At a glance

Generic nameCefazolin PostOperatively
Also known asAncef, Kefzol
SponsorAultman Health Foundation
Drug classFirst-generation cephalosporin
TargetPenicillin-binding proteins (PBPs)
ModalitySmall molecule
Therapeutic areaInfectious Disease
PhaseFDA-approved

Mechanism of action

Cefazolin works by disrupting the cross-linking of peptidoglycan in bacterial cell walls, leading to cell wall instability and bacterial death. It is bactericidal and has broad activity against gram-positive cocci and some gram-negative bacteria. When used postoperatively, it provides prophylaxis against surgical site infections.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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