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Cathflo Activase (Alteplase)

Genentech, Inc. · FDA-approved active Small molecule

Alteplase is a tissue plasminogen activator (tPA) that converts plasminogen to plasmin, which breaks down fibrin clots.

Alteplase is a tissue plasminogen activator (tPA) that converts plasminogen to plasmin, which breaks down fibrin clots. Used for Restoration of function to central venous catheters occluded by thrombus.

At a glance

Generic nameCathflo Activase (Alteplase)
SponsorGenentech, Inc.
Drug classFibrinolytic agent / Tissue plasminogen activator (tPA)
TargetPlasminogen
ModalitySmall molecule
Therapeutic areaCardiovascular / Interventional
PhaseFDA-approved

Mechanism of action

Alteplase is a recombinant human tissue plasminogen activator that directly activates the fibrinolytic system by converting plasminogen to plasmin. Plasmin then degrades fibrin, the structural protein in blood clots, leading to clot dissolution. Cathflo Activase is specifically formulated for catheter-directed thrombolysis to restore patency of occluded central venous catheters.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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