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Carboplatin Injection

Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · FDA-approved active Small molecule

Carboplatin is a platinum-based chemotherapy agent that forms DNA crosslinks, preventing cancer cell replication and inducing apoptosis.

Carboplatin is a platinum-based chemotherapy agent that forms DNA crosslinks, preventing cancer cell replication and inducing apoptosis. Used for Ovarian cancer, Lung cancer, Breast cancer.

At a glance

Generic nameCarboplatin Injection
Also known asCarboplatin, NSC 241240, Carboplatin for injection
SponsorChia Tai Tianqing Pharmaceutical Group Co., Ltd.
Drug classPlatinum-based chemotherapy agent
TargetDNA
ModalitySmall molecule
Therapeutic areaOncology
PhaseFDA-approved

Mechanism of action

Carboplatin binds to DNA and forms interstrand and intrastrand crosslinks, disrupting DNA synthesis and repair mechanisms. This leads to cell cycle arrest and programmed cell death in rapidly dividing cancer cells. It is a second-generation platinum compound with a similar mechanism to cisplatin but with an improved toxicity profile.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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