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captopril, Losartan (drug)

National Taiwan University Hospital · FDA-approved active Small molecule

Captopril and losartan work together to lower blood pressure by inhibiting the renin-angiotensin-aldosterone system through different mechanisms: captopril blocks ACE enzyme while losartan blocks angiotensin II receptor.

Captopril and losartan work together to lower blood pressure by inhibiting the renin-angiotensin-aldosterone system through different mechanisms: captopril blocks ACE enzyme while losartan blocks angiotensin II receptor. Used for Hypertension, Heart failure, Post-myocardial infarction.

At a glance

Generic namecaptopril, Losartan (drug)
SponsorNational Taiwan University Hospital
Drug classACE inhibitor and angiotensin II receptor antagonist combination
TargetACE enzyme and AT1 receptor
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Captopril is an ACE inhibitor that prevents the conversion of angiotensin I to angiotensin II, reducing vasoconstriction and aldosterone secretion. Losartan is an angiotensin II receptor antagonist (ARB) that blocks AT1 receptors, preventing angiotensin II from exerting its vasoconstrictive effects. Together, they provide dual blockade of the renin-angiotensin system for enhanced blood pressure reduction.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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