Last reviewed · How we verify

CAPOXIRI

National Cancer Center Hospital East · Phase 3 active Small molecule

CAPOXIRI is a combination chemotherapy regimen that inhibits DNA synthesis and repair through multiple mechanisms to kill rapidly dividing cancer cells.

CAPOXIRI is a combination chemotherapy regimen that inhibits DNA synthesis and repair through multiple mechanisms to kill rapidly dividing cancer cells. Used for Metastatic colorectal cancer (Phase 3 development).

At a glance

Generic nameCAPOXIRI
Also known asExperimental
SponsorNational Cancer Center Hospital East
Drug classCombination chemotherapy (fluoropyrimidine + platinum agent)
TargetThymidylate synthase (capecitabine); DNA (oxaliplatin cross-linking)
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

CAPOXIRI combines capecitabine (a fluoropyrimidine prodrug converted to 5-FU) with oxaliplatin (a platinum-based alkylating agent). Capecitabine inhibits thymidylate synthase to disrupt DNA synthesis, while oxaliplatin forms DNA cross-links to prevent replication and transcription. Together, these agents provide synergistic cytotoxic activity against colorectal and other solid tumors.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape: