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Canagliflozin (TA-7284)
Canagliflozin (TA-7284) is a SGLT2 inhibitor Small molecule drug developed by Tanabe Pharma Corporation. It is currently FDA-approved for Type 2 diabetes mellitus.
Canagliflozin inhibits sodium-glucose cotransporter 2 (SGLT2) in the kidney, reducing glucose reabsorption and increasing urinary glucose excretion to lower blood glucose levels.
Canagliflozin inhibits sodium-glucose cotransporter 2 (SGLT2) in the kidney, reducing glucose reabsorption and increasing urinary glucose excretion to lower blood glucose levels. Used for Type 2 diabetes mellitus.
At a glance
| Generic name | Canagliflozin (TA-7284) |
|---|---|
| Sponsor | Tanabe Pharma Corporation |
| Drug class | SGLT2 inhibitor |
| Target | SGLT2 (sodium-glucose cotransporter 2) |
| Modality | Small molecule |
| Therapeutic area | Diabetes |
| Phase | FDA-approved |
Mechanism of action
SGLT2 is responsible for reabsorbing filtered glucose in the proximal tubule of the nephron. By blocking this transporter, canagliflozin prevents glucose from being reabsorbed back into the bloodstream, allowing excess glucose to be excreted in the urine. This mechanism is independent of insulin secretion or action, making it effective across different stages of type 2 diabetes.
Approved indications
- Type 2 diabetes mellitus
Common side effects
- Genital mycotic infections
- Urinary tract infections
- Polyuria
- Thirst
- Diabetic ketoacidosis
Key clinical trials
- A Study to Evaluate the PK/PD and Safety of TA-7284 in Patients With Type 2 Diabetes Mellitus Who Have Moderate Renal Impairment (PHASE1)
- Long-Term Safety Study of TA-7284 in Patients With Type 2 Diabetes Mellitus (PHASE3)
- Efficacy and Safety Study of Canagliflozin (TA-7284) in Combination With Insulin in Patients With Type 2 Diabetes Mellitus (PHASE4)
- Long-Term Safety Study of Canagliflozin (TA-7284) in Combination With GLP-1 Analogue in Patients With Type 2 Diabetes Mellitus (PHASE4)
- An Efficacy, Safety, and Tolerability Study for TA-7284 in Patients With Type 2 Diabetes (PHASE2)
- Efficacy and Safety Study of TA-7284 in Patients With Type 2 Diabetes (PHASE3)
- Long-Term Safety Study of Canagliflozin (TA-7284) in Combination With Insulin in Patients With Type 2 Diabetes Mellitus (PHASE4)
- Efficacy and Safety of Canagliflozin (TA-7284) in Patients With Diabetic Nephropathy (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Canagliflozin (TA-7284) CI brief — competitive landscape report
- Canagliflozin (TA-7284) updates RSS · CI watch RSS
- Tanabe Pharma Corporation portfolio CI
Frequently asked questions about Canagliflozin (TA-7284)
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Related
- Drug class: All SGLT2 inhibitor drugs
- Target: All drugs targeting SGLT2 (sodium-glucose cotransporter 2)
- Manufacturer: Tanabe Pharma Corporation — full pipeline
- Therapeutic area: All drugs in Diabetes
- Indication: Drugs for Type 2 diabetes mellitus
- Compare: Canagliflozin (TA-7284) vs similar drugs
- Pricing: Canagliflozin (TA-7284) cost, discount & access