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Calcipotriene/betamethasone

Derm Research, PLLC · FDA-approved active Small molecule

Calcipotriene is a vitamin D analog that regulates skin cell differentiation and proliferation, while betamethasone is a corticosteroid that suppresses inflammation and immune response in the skin.

Calcipotriene is a vitamin D analog that regulates skin cell differentiation and proliferation, while betamethasone is a corticosteroid that suppresses inflammation and immune response in the skin. Used for Plaque psoriasis, Psoriatic dermatitis.

At a glance

Generic nameCalcipotriene/betamethasone
Also known asTaclonex
SponsorDerm Research, PLLC
Drug classVitamin D analog / Corticosteroid combination
TargetVitamin D receptor (VDR) / Glucocorticoid receptor (GR)
ModalitySmall molecule
Therapeutic areaDermatology
PhaseFDA-approved

Mechanism of action

Calcipotriene binds to vitamin D receptors on keratinocytes and immune cells, promoting normal differentiation and reducing excessive proliferation characteristic of psoriasis. Betamethasone acts as a glucocorticoid receptor agonist, rapidly suppressing inflammatory cytokines and immune cell infiltration. Together, they provide complementary anti-inflammatory and anti-proliferative effects on psoriatic plaques.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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