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Bumetanide white, oblong, scored tablet

B&A Therapeutics · Phase 2 active Small molecule

Inhibits the Na-K-2Cl cotransporter 2 (NKCC2) in the thick ascending limb of the loop of Henle.

Inhibits the Na-K-2Cl cotransporter 2 (NKCC2) in the thick ascending limb of the loop of Henle. Used for Edema associated with congestive heart failure, cirrhosis of the liver, and a nephrotic syndrome in adults.

At a glance

Generic nameBumetanide white, oblong, scored tablet
SponsorB&A Therapeutics
Drug classLoop diuretic
TargetNa-K-2Cl cotransporter 2 (NKCC2)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 2

Mechanism of action

This action results in increased excretion of sodium, chloride, potassium, and water, leading to a decrease in blood volume and a subsequent decrease in blood pressure.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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