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Bencycloquidium Bromide Nasal Spray

Yingu Pharmaceutical Co., Ltd · FDA-approved active Small molecule

Bencycloquidium bromide is an anticholinergic agent that blocks muscarinic acetylcholine receptors to reduce nasal secretions and congestion.

Bencycloquidium bromide is an anticholinergic agent that blocks muscarinic acetylcholine receptors to reduce nasal secretions and congestion. Used for Allergic rhinitis with rhinorrhea, Vasomotor rhinitis.

At a glance

Generic nameBencycloquidium Bromide Nasal Spray
Also known asBILITING
SponsorYingu Pharmaceutical Co., Ltd
Drug classAnticholinergic agent
TargetMuscarinic acetylcholine receptor (M3)
ModalitySmall molecule
Therapeutic areaRespiratory / Allergy
PhaseFDA-approved

Mechanism of action

As a quaternary ammonium anticholinergic compound, bencycloquidium bromide antagonizes M3 muscarinic receptors on nasal mucosa, decreasing mucus production and secretion. When delivered as a nasal spray, it provides local anticholinergic effects to alleviate rhinorrhea and nasal congestion associated with allergic rhinitis and other nasal conditions.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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