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Baricitinib Oral Tablet

Azienda Ospedaliero, Universitaria Pisana · Phase 3 active Small molecule

Baricitinib is a JAK inhibitor that blocks Janus kinase signaling to reduce inflammatory cytokine production and immune cell activation.

Baricitinib is a JAK inhibitor that blocks Janus kinase signaling to reduce inflammatory cytokine production and immune cell activation. Used for Rheumatoid arthritis, Atopic dermatitis, Alopecia areata.

At a glance

Generic nameBaricitinib Oral Tablet
Also known asLY3009104, Olumiant, Arm B
SponsorAzienda Ospedaliero, Universitaria Pisana
Drug classJAK inhibitor
TargetJAK1, JAK2
ModalitySmall molecule
Therapeutic areaImmunology
PhasePhase 3

Mechanism of action

Baricitinib selectively inhibits JAK1 and JAK2 enzymes, which are intracellular kinases involved in the signaling of multiple inflammatory cytokines including interferons and interleukins. By blocking JAK-STAT pathway signaling, the drug suppresses the proliferation and activation of immune cells, reducing systemic inflammation and autoimmune responses. This mechanism makes it effective in conditions driven by dysregulated Th1 and Th17 cell responses.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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