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AZD6244 Dosing Period 1

AstraZeneca · Phase 1 active Small molecule

MEK inhibitor

MEK inhibitor Used for Non-small cell lung cancer.

At a glance

Generic nameAZD6244 Dosing Period 1
Also known asAZD6244
SponsorAstraZeneca
Drug classMEK inhibitor
TargetMEK1 and MEK2
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 1

Mechanism of action

AZD6244 is a potent and selective inhibitor of MEK1 and MEK2, enzymes that are key regulators of the MAPK/ERK signaling pathway.

Approved indications

Common side effects

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