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Tecentriq (atezolizumab)
Tecentriq works by blocking a protein called PD-L1, which helps cancer cells hide from the immune system.
Tecentriq (atezolizumab) is a programmed death receptor-1 blocking antibody developed by Genentech Inc. It targets the programmed cell death 1 ligand 1, a protein that can help cancer cells evade the immune system. Tecentriq is approved to treat various types of cancer, including lung, breast, liver, and bladder cancers. The drug has a half-life of 27 days and is still patented. Key safety considerations include immune-mediated reactions and infusion-related reactions.
At a glance
| Generic name | atezolizumab |
|---|---|
| Sponsor | Roche |
| Drug class | Programmed Death Receptor-1 Blocking Antibody [EPC] |
| Target | Programmed cell death 1 ligand 1 |
| Modality | Monoclonal antibody |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
| First approval | 2016 |
| Annual revenue | 3700 |
Mechanism of action
PD-L1 may be expressed on tumor cells and/or tumor infiltrating immune cells and can contribute to the inhibition of the anti-tumor immune response in the tumor microenvironment. Binding of PD-L1 to the PD-1 and B7.1 receptors found on cells and antigen presenting cells suppresses cytotoxic T-cell activity, T-cell proliferation and cytokine production.Atezolizumab is monoclonal antibody that binds to PD-L1 and blocks its interactions with both PD-1 and B7.1 receptors. This releases the PD-L1/PD-1 mediated inhibition of the immune response, including activation of the anti-tumor immune response without inducing antibody-dependent cellular cytotoxicity. In syngeneic mouse tumor models, blocking PD-L1 activity resulted in decreased tumor growth.In mouse models of cancer, dual inhibition of the PD-1/PD-L1 and MAPK pathways suppresses tumor growth and improves tumor immunogenicity through increased antigen presentation and cell infiltration and activation compared t
Approved indications
- Extensive stage primary small cell carcinoma of lung
- Germline BRCA-mutated, HER2-negative metastatic breast cancer
- Liver cell carcinoma
- Metastatic non-small cell lung cancer
- Transitional cell carcinoma
Common side effects
- Fatigue/asthenia
- Fatigue
- Nausea
- Alopecia
- Constipation
- Diarrhea
- Decreased appetite
- Cough
- Dyspnea
- Hypertension
- Proteinuria
- Rash
Key clinical trials
- A Study of Atezolizumab in Combination With Bevacizumab Compared With Sorafenib in Patients With Untreated Locally Advanced or Metastatic Hepatocellular Carcinoma (PHASE3)
- A Study of Atezolizumab in Participants With Locally Advanced or Metastatic Urothelial Bladder Cancer (Cohort 1) (PHASE2)
- A Study of Atezolizumab in Combination With Carboplatin Plus (+) Paclitaxel With or Without Bevacizumab Compared With Carboplatin+Paclitaxel+Bevacizumab in Participants With Stage IV Non-Squamous Non-Small Cell Lung Cancer (NSCLC) (PHASE3)
- A Study of Atezolizumab (MPDL3280A) Compared With a Platinum Agent (Cisplatin or Carboplatin) + (Pemetrexed or Gemcitabine) in Participants With Stage IV Non-Squamous or Squamous Non-Small Cell Lung Cancer (NSCLC) [IMpower110] (PHASE3)
- A Study of Carboplatin Plus Etoposide With or Without Atezolizumab in Participants With Untreated Extensive-Stage (ES) Small Cell Lung Cancer (SCLC) (PHASE3)
- A Study of Atezolizumab Plus Cobimetinib and Vemurafenib Versus Placebo Plus Cobimetinib and Vemurafenib in Previously Untreated BRAFv600 Mutation-Positive Patients With Metastatic or Unresectable Locally Advanced Melanoma (PHASE3)
- A Study of Atezolizumab Compared With Docetaxel in Participants With Locally Advanced or Metastatic Non-Small Cell Lung Cancer Who Have Failed Platinum-Containing Therapy (PHASE3)
- A Study of Atezolizumab in Combination With Carboplatin Plus (+) Nab-Paclitaxel Compared With Carboplatin+Nab-Paclitaxel in Participants With Stage IV Non-Squamous Non-Small Cell Lung Cancer (NSCLC) (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
| SEC EDGAR | Revenue + earnings |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Tecentriq CI brief — competitive landscape report
- Tecentriq updates RSS · CI watch RSS
- Roche portfolio CI