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Atenolol/HCTZ/Trandolapril
Atenolol/HCTZ/Trandolapril is a Antihypertensive combination (beta-blocker/thiazide diuretic/ACE inhibitor) Small molecule drug developed by University of Florida. It is currently FDA-approved for Hypertension.
This triple-combination antihypertensive reduces blood pressure through three complementary mechanisms: beta-blockade, diuresis, and ACE inhibition.
This triple-combination antihypertensive reduces blood pressure through three complementary mechanisms: beta-blockade, diuresis, and ACE inhibition. Used for Hypertension.
At a glance
| Generic name | Atenolol/HCTZ/Trandolapril |
|---|---|
| Sponsor | University of Florida |
| Drug class | Antihypertensive combination (beta-blocker/thiazide diuretic/ACE inhibitor) |
| Target | Beta-1 adrenergic receptor, sodium-chloride cotransporter, angiotensin-converting enzyme |
| Modality | Small molecule |
| Therapeutic area | Cardiovascular |
| Phase | FDA-approved |
Mechanism of action
Atenolol is a beta-1 selective antagonist that reduces heart rate and cardiac contractility. Hydrochlorothiazide (HCTZ) is a thiazide diuretic that decreases blood volume and sodium reabsorption. Trandolapril is an ACE inhibitor that blocks angiotensin II formation, reducing vasoconstriction and aldosterone secretion. Together, these agents provide synergistic blood pressure reduction.
Approved indications
- Hypertension
Common side effects
- Fatigue
- Dizziness
- Cough
- Hyperglycemia
- Hypokalemia
- Bradycardia
- Erectile dysfunction
Key clinical trials
- ACEI or ARB and COVID-19 Severity and Mortality in US Veterans
- INVEST: INternational VErapamil SR Trandolapril STudy (PHASE4)
- Renin-Guided Therapeutics in the Management of Untreated, Uncontrolled, or Complicated Hypertension (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Atenolol/HCTZ/Trandolapril CI brief — competitive landscape report
- Atenolol/HCTZ/Trandolapril updates RSS · CI watch RSS
- University of Florida portfolio CI
Frequently asked questions about Atenolol/HCTZ/Trandolapril
What is Atenolol/HCTZ/Trandolapril?
How does Atenolol/HCTZ/Trandolapril work?
What is Atenolol/HCTZ/Trandolapril used for?
Who makes Atenolol/HCTZ/Trandolapril?
What drug class is Atenolol/HCTZ/Trandolapril in?
What development phase is Atenolol/HCTZ/Trandolapril in?
What are the side effects of Atenolol/HCTZ/Trandolapril?
What does Atenolol/HCTZ/Trandolapril target?
Related
- Drug class: All Antihypertensive combination (beta-blocker/thiazide diuretic/ACE inhibitor) drugs
- Target: All drugs targeting Beta-1 adrenergic receptor, sodium-chloride cotransporter, angiotensin-converting enzyme
- Manufacturer: University of Florida — full pipeline
- Therapeutic area: All drugs in Cardiovascular
- Indication: Drugs for Hypertension
- Compare: Atenolol/HCTZ/Trandolapril vs similar drugs
- Pricing: Atenolol/HCTZ/Trandolapril cost, discount & access