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aspart insulin or lipro insulin

Nanjing First Hospital, Nanjing Medical University · FDA-approved active Small molecule

Aspart insulin is a rapid-acting insulin analog that binds to insulin receptors to promote glucose uptake and utilization in peripheral tissues.

Aspart insulin is a rapid-acting insulin analog that binds to insulin receptors to promote glucose uptake and utilization in peripheral tissues. Used for Type 1 diabetes mellitus, Type 2 diabetes mellitus.

At a glance

Generic nameaspart insulin or lipro insulin
SponsorNanjing First Hospital, Nanjing Medical University
Drug classRapid-acting insulin analog
TargetInsulin receptor
ModalitySmall molecule
Therapeutic areaDiabetes
PhaseFDA-approved

Mechanism of action

Aspart insulin is a recombinant human insulin analog with a single amino acid substitution (aspartic acid at position B28) that allows faster absorption and onset of action compared to regular human insulin. It binds to the insulin receptor on muscle, fat, and liver cells to facilitate glucose transport into cells and promote anabolic metabolism, effectively lowering blood glucose levels in diabetic patients.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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