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Aripiprazole/Escitalopram combination

Massachusetts General Hospital · FDA-approved active Small molecule

This combination uses aripiprazole (a dopamine D2 receptor partial agonist) and escitalopram (a selective serotonin reuptake inhibitor) to modulate both dopaminergic and serotonergic neurotransmission for psychiatric symptom management.

This combination uses aripiprazole (a dopamine D2 receptor partial agonist) and escitalopram (a selective serotonin reuptake inhibitor) to modulate both dopaminergic and serotonergic neurotransmission for psychiatric symptom management. Used for Schizophrenia with comorbid depression, Bipolar disorder with depressive symptoms, Major depressive disorder with psychotic features.

At a glance

Generic nameAripiprazole/Escitalopram combination
Also known asAbilify/ Lexapro
SponsorMassachusetts General Hospital
Drug classAtypical antipsychotic and selective serotonin reuptake inhibitor combination
TargetDopamine D2 receptor (partial agonist), serotonin 5-HT1A receptor (partial agonist), serotonin transporter (SERT inhibitor)
ModalitySmall molecule
Therapeutic areaPsychiatry
PhaseFDA-approved

Mechanism of action

Aripiprazole acts as a partial agonist at dopamine D2 receptors and serotonin 5-HT1A receptors, stabilizing dopamine signaling in psychotic and mood disorders. Escitalopram inhibits serotonin reuptake, increasing synaptic serotonin availability. Together, they address both psychotic symptoms and comorbid depression or anxiety.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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