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Aripiprazole 8-week group

Seoul National University Hospital · FDA-approved active Small molecule

Aripiprazole is a dopamine D2/D3 receptor partial agonist that modulates dopaminergic and serotonergic neurotransmission to treat psychotic and mood disorders.

Aripiprazole is a dopamine D2/D3 receptor partial agonist that modulates dopaminergic and serotonergic neurotransmission to treat psychotic and mood disorders. Used for Schizophrenia, Bipolar I disorder (acute manic or mixed episodes), Major depressive disorder (adjunctive treatment).

At a glance

Generic nameAripiprazole 8-week group
Also known asAbilify®
SponsorSeoul National University Hospital
Drug classAtypical antipsychotic
TargetDopamine D2/D3 receptor (partial agonist); serotonin 5-HT1A receptor
ModalitySmall molecule
Therapeutic areaPsychiatry
PhaseFDA-approved

Mechanism of action

Aripiprazole acts as a partial agonist at dopamine D2 and D3 receptors, providing dopaminergic stabilization rather than pure antagonism. This mechanism reduces excessive dopamine signaling in hyperactive pathways while maintaining adequate dopamine function in hypoactive pathways. It also has activity at serotonin 5-HT1A and 5-HT7 receptors, contributing to its efficacy in treating schizophrenia, bipolar disorder, and depression.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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