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Apremilast Modified Release 13

Amgen · Phase 1 active Small molecule

Apremilast is a small molecule inhibitor of phosphodiesterase 4 (PDE4), which leads to increased intracellular levels of cyclic adenosine monophosphate (cAMP).

Apremilast is a small molecule inhibitor of phosphodiesterase 4 (PDE4), which leads to increased intracellular levels of cyclic adenosine monophosphate (cAMP). Used for Plaque psoriasis, Psoriatic arthritis.

At a glance

Generic nameApremilast Modified Release 13
SponsorAmgen
Drug classPDE4 inhibitor
TargetPDE4
ModalitySmall molecule
Therapeutic areaImmunology
PhasePhase 1

Mechanism of action

By inhibiting PDE4, apremilast reduces the production of pro-inflammatory mediators and increases the production of anti-inflammatory mediators, thereby modulating the immune response and reducing inflammation.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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