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Amzeeq 4% Topical Foam

Edward Lain, MD · FDA-approved active Small molecule

Amzeeq is a topical foam formulation of minocycline that reduces inflammation and bacterial colonization in acne by inhibiting bacterial protein synthesis and suppressing inflammatory mediators.

Amzeeq is a topical foam formulation of minocycline that reduces inflammation and bacterial colonization in acne by inhibiting bacterial protein synthesis and suppressing inflammatory mediators. Used for Acne vulgaris.

At a glance

Generic nameAmzeeq 4% Topical Foam
Also known asminocycline
SponsorEdward Lain, MD
Drug classTetracycline antibiotic
TargetBacterial 30S ribosomal subunit; matrix metalloproteinases
ModalitySmall molecule
Therapeutic areaDermatology
PhaseFDA-approved

Mechanism of action

Minocycline is a tetracycline antibiotic that penetrates sebaceous follicles and exerts both antimicrobial effects against Cutibacterium acnes and anti-inflammatory effects by inhibiting matrix metalloproteinases and reducing cytokine production. The foam formulation provides enhanced penetration and cosmetic acceptability for topical delivery to acne-prone skin.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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