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Amlodipine/Olmesartan

Radboud University Medical Center · FDA-approved active Small molecule

Amlodipine relaxes blood vessels by blocking calcium channels, while olmesartan blocks angiotensin II receptors to reduce vasoconstriction and lower blood pressure.

Amlodipine relaxes blood vessels by blocking calcium channels, while olmesartan blocks angiotensin II receptors to reduce vasoconstriction and lower blood pressure. Used for Hypertension.

At a glance

Generic nameAmlodipine/Olmesartan
SponsorRadboud University Medical Center
Drug classCalcium channel blocker / Angiotensin II receptor blocker combination
TargetL-type calcium channels (amlodipine); AT1 angiotensin II receptor (olmesartan)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Amlodipine is a dihydropyridine calcium channel blocker that inhibits L-type calcium channels in vascular smooth muscle, causing vasodilation. Olmesartan is an angiotensin II receptor blocker (ARB) that antagonizes AT1 receptors, preventing angiotensin II-mediated vasoconstriction and aldosterone release. Together, these complementary mechanisms provide additive antihypertensive effects.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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