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Amlodipine Besylate / Benazepril Hydrochloride

Dr. Reddy's Laboratories Limited · FDA-approved active Small molecule

Amlodipine Besylate / Benazepril Hydrochloride is a Calcium channel blocker / ACE inhibitor combination Small molecule drug developed by Dr. Reddy's Laboratories Limited. It is currently FDA-approved for Hypertension. Also known as: Lotrel® (10 mg Amlodipine Besylate / 20 mg Benazepril, Hydrochloride Capsules).

This combination drug lowers blood pressure by relaxing blood vessels (amlodipine) and reducing angiotensin II production (benazepril).

This combination drug lowers blood pressure by relaxing blood vessels (amlodipine) and reducing angiotensin II production (benazepril). Used for Hypertension.

At a glance

Generic nameAmlodipine Besylate / Benazepril Hydrochloride
Also known asLotrel® (10 mg Amlodipine Besylate / 20 mg Benazepril, Hydrochloride Capsules)
SponsorDr. Reddy's Laboratories Limited
Drug classCalcium channel blocker / ACE inhibitor combination
TargetL-type calcium channels; Angiotensin-converting enzyme (ACE)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Amlodipine is a calcium channel blocker that prevents calcium from entering vascular smooth muscle cells, causing vasodilation. Benazepril is an ACE inhibitor that blocks the conversion of angiotensin I to angiotensin II, a potent vasoconstrictor, thereby reducing peripheral vascular resistance and blood pressure. Together, these complementary mechanisms provide additive antihypertensive effects.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Amlodipine Besylate / Benazepril Hydrochloride

What is Amlodipine Besylate / Benazepril Hydrochloride?

Amlodipine Besylate / Benazepril Hydrochloride is a Calcium channel blocker / ACE inhibitor combination drug developed by Dr. Reddy's Laboratories Limited, indicated for Hypertension.

How does Amlodipine Besylate / Benazepril Hydrochloride work?

This combination drug lowers blood pressure by relaxing blood vessels (amlodipine) and reducing angiotensin II production (benazepril).

What is Amlodipine Besylate / Benazepril Hydrochloride used for?

Amlodipine Besylate / Benazepril Hydrochloride is indicated for Hypertension.

Who makes Amlodipine Besylate / Benazepril Hydrochloride?

Amlodipine Besylate / Benazepril Hydrochloride is developed and marketed by Dr. Reddy's Laboratories Limited (see full Dr. Reddy's Laboratories Limited pipeline at /company/dr-reddy-s-laboratories-limited).

Is Amlodipine Besylate / Benazepril Hydrochloride also known as anything else?

Amlodipine Besylate / Benazepril Hydrochloride is also known as Lotrel® (10 mg Amlodipine Besylate / 20 mg Benazepril, Hydrochloride Capsules).

What drug class is Amlodipine Besylate / Benazepril Hydrochloride in?

Amlodipine Besylate / Benazepril Hydrochloride belongs to the Calcium channel blocker / ACE inhibitor combination class. See all Calcium channel blocker / ACE inhibitor combination drugs at /class/calcium-channel-blocker-ace-inhibitor-combination.

What development phase is Amlodipine Besylate / Benazepril Hydrochloride in?

Amlodipine Besylate / Benazepril Hydrochloride is FDA-approved (marketed).

What are the side effects of Amlodipine Besylate / Benazepril Hydrochloride?

Common side effects of Amlodipine Besylate / Benazepril Hydrochloride include Headache, Dizziness, Fatigue, Peripheral edema, Cough, Hyperkalemia.

What does Amlodipine Besylate / Benazepril Hydrochloride target?

Amlodipine Besylate / Benazepril Hydrochloride targets L-type calcium channels; Angiotensin-converting enzyme (ACE) and is a Calcium channel blocker / ACE inhibitor combination.

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