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Alogliptin and insulin
Alogliptin and insulin is a DPP-4 inhibitor combined with insulin Small molecule drug developed by Takeda. It is currently in Phase 3 development for Type 2 diabetes mellitus in patients inadequately controlled on insulin alone. Also known as: alogliptin, SYR110322.
Alogliptin inhibits dipeptidyl peptidase-4 (DPP-4) to increase incretin levels and improve glucose control, while insulin provides exogenous glucose-lowering activity.
Alogliptin inhibits dipeptidyl peptidase-4 (DPP-4) to increase incretin levels and improve glucose control, while insulin provides exogenous glucose-lowering activity. Used for Type 2 diabetes mellitus in patients inadequately controlled on insulin alone.
At a glance
| Generic name | Alogliptin and insulin |
|---|---|
| Also known as | alogliptin, SYR110322 |
| Sponsor | Takeda |
| Drug class | DPP-4 inhibitor combined with insulin |
| Target | DPP-4 (dipeptidyl peptidase-4) |
| Modality | Small molecule |
| Therapeutic area | Diabetes |
| Phase | Phase 3 |
Mechanism of action
Alogliptin is a DPP-4 inhibitor that prevents the degradation of glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP), thereby enhancing insulin secretion and reducing glucagon in response to elevated blood glucose. The combination with insulin provides additional glycemic control through exogenous insulin replacement, targeting both endogenous and exogenous pathways of glucose homeostasis in type 2 diabetes.
Approved indications
- Type 2 diabetes mellitus in patients inadequately controlled on insulin alone
Common side effects
- Hypoglycemia
- Nasopharyngitis
- Upper respiratory tract infection
- Headache
- Pancreatitis
Key clinical trials
- Comparative Effectiveness and Safety of Four Second Line Pharmacological Strategies in Type 2 Diabetes Study
- A Study for Comparison of Canagliflozin Versus Alternative Antihyperglycemic Treatments on Risk of Heart Failure Hospitalization and Amputation for Participants With Type 2 Diabetes Mellitus and the Subpopulation With Established Cardiovascular Disease
- Safety of Sodium-glucose Cotransporter 2 (SGLT2) Inhibitors Among Patients with Type 2 Diabetes
- Real-World Evaluation of Omarigliptin for Type 2 Diabetes Meliitus in Bangladesh (PHASE4)
- Gliflozins and Cardiovascular Risk Factors in Type 2 Diabetes (GIOIA)
- BESTMED: Observational Evaluation of Second Line Therapy Medications in Diabetes
- Phase 3 Alogliptin Pediatric Study (PHASE3)
- The Effect of Alogliptin on Pulmonary Function in Obese Patients With Type 2 Diabetes Inadequately Controlled by Metformin Monotherapy (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Alogliptin and insulin CI brief — competitive landscape report
- Alogliptin and insulin updates RSS · CI watch RSS
- Takeda portfolio CI
Frequently asked questions about Alogliptin and insulin
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Related
- Drug class: All DPP-4 inhibitor combined with insulin drugs
- Target: All drugs targeting DPP-4 (dipeptidyl peptidase-4)
- Manufacturer: Takeda — full pipeline
- Therapeutic area: All drugs in Diabetes
- Indication: Drugs for Type 2 diabetes mellitus in patients inadequately controlled on insulin alone
- Also known as: alogliptin, SYR110322
- Compare: Alogliptin and insulin vs similar drugs
- Pricing: Alogliptin and insulin cost, discount & access