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AGN-210961 Formulation 5

Allergan · Phase 2 active Small molecule

AGN-210961 Formulation 5 is a medication that targets the PCSK9 protein to lower LDL cholesterol.

AGN-210961 Formulation 5 is a medication that targets the PCSK9 protein to lower LDL cholesterol. Used for Hypercholesterolemia.

At a glance

Generic nameAGN-210961 Formulation 5
SponsorAllergan
Drug classPCSK9 inhibitor
TargetPCSK9
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 2

Mechanism of action

By binding to PCSK9, AGN-210961 Formulation 5 inhibits the degradation of LDL receptors, leading to increased clearance of LDL cholesterol from the bloodstream. This results in a reduction of LDL cholesterol levels in the blood, which can help to slow the progression of atherosclerotic cardiovascular disease.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results