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Adjuvant tislelizumab plus lenvatinib

Guangxi Medical University · Phase 3 active Small molecule

Adjuvant tislelizumab plus lenvatinib is a PD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination Small molecule drug developed by Guangxi Medical University. It is currently in Phase 3 development for Adjuvant treatment of hepatocellular carcinoma (Phase 3).

Tislelizumab blocks PD-1 on immune cells to enhance anti-tumor immunity, while lenvatinib inhibits multiple receptor tyrosine kinases to suppress tumor angiogenesis and growth.

Tislelizumab blocks PD-1 on immune cells to enhance anti-tumor immunity, while lenvatinib inhibits multiple receptor tyrosine kinases to suppress tumor angiogenesis and growth. Used for Adjuvant treatment of hepatocellular carcinoma (Phase 3).

At a glance

Generic nameAdjuvant tislelizumab plus lenvatinib
SponsorGuangxi Medical University
Drug classPD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination
TargetPD-1 (tislelizumab); FGFR, VEGFR, RET, KIT (lenvatinib)
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

Tislelizumab is a humanized anti-PD-1 monoclonal antibody that restores T-cell-mediated immune responses against cancer cells. Lenvatinib is a multi-targeted tyrosine kinase inhibitor that blocks FGFR, VEGFR, RET, and KIT signaling, reducing tumor vascularity and proliferation. The combination leverages immunotherapy with targeted anti-angiogenic therapy to enhance overall anti-tumor efficacy.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Adjuvant tislelizumab plus lenvatinib

What is Adjuvant tislelizumab plus lenvatinib?

Adjuvant tislelizumab plus lenvatinib is a PD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination drug developed by Guangxi Medical University, indicated for Adjuvant treatment of hepatocellular carcinoma (Phase 3).

How does Adjuvant tislelizumab plus lenvatinib work?

Tislelizumab blocks PD-1 on immune cells to enhance anti-tumor immunity, while lenvatinib inhibits multiple receptor tyrosine kinases to suppress tumor angiogenesis and growth.

What is Adjuvant tislelizumab plus lenvatinib used for?

Adjuvant tislelizumab plus lenvatinib is indicated for Adjuvant treatment of hepatocellular carcinoma (Phase 3).

Who makes Adjuvant tislelizumab plus lenvatinib?

Adjuvant tislelizumab plus lenvatinib is developed by Guangxi Medical University (see full Guangxi Medical University pipeline at /company/guangxi-medical-university).

What drug class is Adjuvant tislelizumab plus lenvatinib in?

Adjuvant tislelizumab plus lenvatinib belongs to the PD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination class. See all PD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination drugs at /class/pd-1-inhibitor-multi-targeted-tyrosine-kinase-inhibitor-combination.

What development phase is Adjuvant tislelizumab plus lenvatinib in?

Adjuvant tislelizumab plus lenvatinib is in Phase 3.

What are the side effects of Adjuvant tislelizumab plus lenvatinib?

Common side effects of Adjuvant tislelizumab plus lenvatinib include Fatigue, Hypertension, Diarrhea, Decreased appetite, Immune-related adverse events (e.g., hepatitis, pneumonitis), Proteinuria.

What does Adjuvant tislelizumab plus lenvatinib target?

Adjuvant tislelizumab plus lenvatinib targets PD-1 (tislelizumab); FGFR, VEGFR, RET, KIT (lenvatinib) and is a PD-1 inhibitor + multi-targeted tyrosine kinase inhibitor combination.

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