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ACTIQ®

Cephalon · Phase 2 active Small molecule

ACTIQ® delivers fentanyl, a potent opioid analgesic, directly to the oral mucosa for rapid absorption and pain relief.

ACTIQ® delivers fentanyl, a potent opioid analgesic, directly to the oral mucosa for rapid absorption and pain relief. Used for Breakthrough cancer pain in adults who are already receiving and who are tolerant to around-the-clock opioid therapy for their underlying persistent cancer pain.

At a glance

Generic nameACTIQ®
SponsorCephalon
Drug classopioid analgesic
Targetmu-opioid receptors
ModalitySmall molecule
Therapeutic areaPain Management
PhasePhase 2

Mechanism of action

Fentanyl acts by binding to the mu-opioid receptors in the central nervous system, which leads to a decrease in the perception of pain and an increase in pain tolerance.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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