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Aclidinium Bromide 400 µg

AstraZeneca · Phase 3 active Small molecule

Aclidinium bromide is a muscarinic M3 receptor antagonist that blocks acetylcholine signaling in airway smooth muscle, causing bronchodilation.

Aclidinium bromide is a muscarinic M3 receptor antagonist that blocks acetylcholine signaling in airway smooth muscle, causing bronchodilation. Used for Chronic obstructive pulmonary disease (COPD) maintenance treatment.

At a glance

Generic nameAclidinium Bromide 400 µg
SponsorAstraZeneca
Drug classLong-acting muscarinic antagonist (LAMA)
TargetMuscarinic M3 receptor
ModalitySmall molecule
Therapeutic areaRespiratory
PhasePhase 3

Mechanism of action

Aclidinium is a long-acting anticholinergic (LAMA) that selectively antagonizes M3 muscarinic receptors on airway smooth muscle and mucus glands. By blocking acetylcholine-mediated bronchoconstriction, it produces sustained airway relaxation and improved airflow. The drug is rapidly hydrolyzed by non-specific esterases, minimizing systemic anticholinergic effects.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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