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Acetazolamide first, then Furosemide

Rabin Medical Center · Phase 1 active Small molecule

Acetazolamide inhibits carbonic anhydrase, reducing the formation of bicarbonate ions and increasing urinary excretion of sodium, potassium, and water.

Acetazolamide inhibits carbonic anhydrase, reducing the formation of bicarbonate ions and increasing urinary excretion of sodium, potassium, and water. Used for Glaucoma, Edema, Seizures.

At a glance

Generic nameAcetazolamide first, then Furosemide
SponsorRabin Medical Center
Drug classCarbonic anhydrase inhibitor
TargetCarbonic anhydrase
ModalitySmall molecule
Therapeutic areaOphthalmology
PhasePhase 1

Mechanism of action

By inhibiting carbonic anhydrase, acetazolamide decreases the reabsorption of bicarbonate in the renal tubules, leading to increased excretion of bicarbonate, sodium, and water, which can help reduce intraocular pressure and treat glaucoma or edema.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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